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Michael D Edstein Selected Research

Oral Administration

10/2019Development of pyridyl thiosemicarbazones as highly potent agents for the treatment of malaria after oral administration.
1/20193,3'-Disubstituted 5,5'-Bi(1,2,4-triazine) Derivatives with Potent in Vitro and in Vivo Antimalarial Activity.

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Michael D Edstein Research Topics

Disease

29Malaria
10/2022 - 09/2003
15Infections
10/2022 - 09/2003
15Falciparum Malaria (Plasmodium falciparum Malaria)
10/2022 - 07/2002
6Vivax Malaria
01/2019 - 06/2006
4Parasitemia
06/2022 - 09/2015
4Body Weight (Weight, Body)
01/2018 - 08/2009
2Hemolysis
10/2022 - 01/2005
1Acute Kidney Injury (Acute Renal Failure)
10/2022
1Carcinoma (Carcinomatosis)
07/2021
1Parasitic Diseases (Parasitic Disease)
01/2018
1Vector Borne Diseases
10/2016
1Abdominal Pain (Pain, Abdominal)
10/2011
1Sleep Initiation and Maintenance Disorders (Insomnia)
10/2011
1Headache (Headaches)
10/2011
1Nausea
10/2011
1Bites and Stings (Sting)
02/2010

Drug/Important Bio-Agent (IBA)

14Antimalarials (Antimalarial Agents)IBA
01/2021 - 09/2003
10ArtesunateIBA
10/2021 - 12/2005
10artemisinin (artemisinine)IBA
01/2020 - 05/2009
9Chloroquine (Aralen)FDA LinkGeneric
10/2021 - 07/2002
9Pharmaceutical PreparationsIBA
01/2020 - 01/2005
8piperaquineIBA
06/2022 - 02/2009
7tafenoquineIBA
06/2022 - 12/2003
6artenimol (dihydroartemisinin)IBA
01/2019 - 02/2009
5Mefloquine (Lariam)FDA LinkGeneric
01/2016 - 02/2005
5PrimaquineFDA Link
06/2007 - 01/2005
4JPC-3210IBA
01/2020 - 01/2016
3Amodiaquine (Camoquin)FDA Link
01/2018 - 05/2009
2ProdrugsIBA
07/2021 - 09/2015
2Drug CombinationsIBA
01/2020 - 03/2015
2pyrimethamine drug combination fanasil (Fansidar)FDA Link
03/2006 - 09/2003
1Acetaminophen (Paracetamol)FDA LinkGeneric
10/2022
1CreatinineIBA
10/2022
1Hemoglobins (Hemoglobin)IBA
10/2022
1EnzymesIBA
02/2022
1AntigensIBA
02/2022
1ImmunosorbentsIBA
02/2022
1AntibodiesIBA
02/2022
1phosphoramidic acidIBA
07/2021
1TriazinesIBA
01/2021
1QuinolonesIBA
01/2020
1ThiosemicarbazonesIBA
10/2019
1LumefantrineFDA Link
01/2019
1ArtemetherFDA Link
01/2019
1Azithromycin (Zithromax)FDA LinkGeneric
07/2016
1pyridineIBA
01/2016
1Phenol (Carbolic Acid)FDA Link
01/2016
1VaccinesIBA
01/2016
1alpha- 2- pyridinyl- 2,8- bis(trifluoromethyl)- 4- quinolinemethanolIBA
01/2016
1pyrimidineIBA
01/2016
1thiaplakortone AIBA
02/2014
1halofantrine (Halfan)FDA Link
11/2012
1Proteins (Proteins, Gene)FDA Link
02/2010
1artemisoneIBA
08/2009
1thymidylate synthase-dihydrofolate reductaseIBA
10/2007
1A-factor (Streptomyces)IBA
06/2006
1Doxycycline (Periostat)FDA LinkGeneric
02/2005
1Mannich BasesIBA
01/2005
1Oxidoreductases (Dehydrogenase)IBA
01/2005
1Glucose (Dextrose)FDA LinkGeneric
01/2005

Therapy/Procedure

7Therapeutics
01/2020 - 09/2003
2Oral Administration
10/2019 - 01/2019
1Chemoprevention
01/2005
1Drug Therapy (Chemotherapy)
09/2003